@<TRIPOS>COMMENTLIGANDBOX_ID = HTS2204-01076016-01 SOURCE = Namiki2204 SOURCE_ID = NS-007347376-0000 MOLECULAR_FORMULA = C13H13N2O3Br MOLECULAR_WEIGHT = 325.162 MOLECULAR_CHARGE = 0 NUM_OF_DONOR = 1 NUM_OF_ACCEPTOR = 3 NUM_OF_CHIRAL_ATOMS = 0 TPSA = 60.3300 HOMO = -8.6798 LUMO = -0.1426 mLOGS = -4.032 mLOGD = 2.518 mLOGPA = -5.049@<TRIPOS>MOLECULEHTS2204-01076016-01 32 33 0 0 0 SMALL MOPAC_AM1BCC@<TRIPOS>ATOM1 N1 6.4090 4.1990 -1.3300 N.ar 1 LGD -0.0939 2 C1 6.4680 2.9720 -0.7000 C.ar 1 LGD -0.0172 3 C2 5.9290 3.9700 -2.6370 C.ar 1 LGD -0.0932 4 C3 6.0510 1.9900 -1.5450 C.ar 1 LGD -0.0954 5 C4 5.6940 2.6040 -2.7970 C.ar 1 LGD -0.1843 6 C5 6.8470 5.4900 -0.7720 C.3 1 LGD -0.0027 7 C6 8.3670 5.6570 -0.8290 C.2 1 LGD 0.6456 8 C7 6.8880 2.7000 0.6100 C.ar 1 LGD -0.1547 9 C8 11.1270 4.7320 1.5930 C.2 1 LGD 0.6282 10 C9 6.0200 0.6460 -1.1550 C.ar 1 LGD -0.0465 11 N2 9.1050 5.3510 0.3020 N.am 1 LGD -0.5953 12 O1 8.9350 6.0390 -1.8380 O.2 1 LGD -0.5756 13 O2 10.4490 4.4660 2.5740 O.2 1 LGD -0.5338 14 C10 10.5730 5.3360 0.2980 C.3 1 LGD 0.0634 15 C11 6.4390 0.3340 0.1550 C.ar 1 LGD -0.0469 16 C12 6.8710 1.3550 1.0350 C.ar 1 LGD -0.0828 17 O3 12.4740 4.5250 1.5020 O.3 1 LGD -0.4265 18 Br1 6.4220 -1.4820 0.7450 Br 1 LGD -0.1068 19 C13 13.1690 3.9540 2.6270 C.3 1 LGD 0.1298 20 H1 5.8010 4.7790 -3.3450 H 1 LGD 0.1742 21 H2 5.3260 2.1260 -3.6980 H 1 LGD 0.1637 22 H3 6.3860 6.3070 -1.3410 H 1 LGD 0.0804 23 H4 6.5170 5.5670 0.2710 H 1 LGD 0.0804 24 H5 7.2150 3.4880 1.2810 H 1 LGD 0.1332 25 H6 5.6860 -0.1290 -1.8400 H 1 LGD 0.1515 26 H7 8.6230 5.0640 1.1420 H 1 LGD 0.3310 27 H8 10.9660 6.3550 0.1940 H 1 LGD 0.0866 28 H9 10.9410 4.7350 -0.5440 H 1 LGD 0.0866 29 H10 7.1910 1.1040 2.0420 H 1 LGD 0.1474 30 H11 12.7580 2.9650 2.8660 H 1 LGD 0.0512 31 H12 14.2350 3.8440 2.3910 H 1 LGD 0.0512 32 H13 13.0690 4.6030 3.5060 H 1 LGD 0.0512@<TRIPOS>BOND1 1 2 1 2 1 3 1 3 2 4 ar 4 3 5 2 5 1 6 1 6 6 7 1 7 2 8 ar 8 9 14 1 9 4 10 ar 10 7 11 am 11 7 12 2 12 9 13 2 13 11 14 1 14 15 16 ar 15 8 16 ar 16 9 17 1 17 15 18 1 18 17 19 1 19 4 5 1 20 10 15 ar 21 3 20 1 22 5 21 1 23 6 22 1 24 6 23 1 25 8 24 1 26 10 25 1 27 11 26 1 28 14 27 1 29 14 28 1 30 16 29 1 31 19 30 1 32 19 31 1 33 19 32 1